Synthesis and sulfatase inhibitory activities of non-steroidal estrone sulfatase inhibitors

Biological Aromatization of Steroids

Kenneth J. Ryan · Journal of Biological Chemistry · 1959 · 595 citations · Full text

Life Sciences, Biochemistry, Pharmacology +12

In Situ Estrogen Production via the Estrone Sulfatase Pathway in Breast Tumors: Relative Importance versus the Aromatase Pathway*

Steven J. Santner, Peter D. Feil, Richard J. Santen · The Journal of Clinical Endocrinology & Metabolism · 1984 · 406 citations

Life Sciences, Biochemistry, Oncology +17

Estrone sulfamates: potent inhibitors of estrone sulfatase with therapeutic potential

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Effects of Plasma Estrogen Sulfates in Mammary Cancer Cells*

Françoise Vignon, M. Terqui, B R Westley et al. · Endocrinology · 1980 · 178 citations

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Inactivation of Steroid Sulfatase by an Active Site-Directed Inhibitor, Estrone-3-O-Sulfamate

Atul Purohit, Gary J. Williams, Nicola M. Howarth et al. · Biochemistry · 1995 · 170 citations

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