Concepedia

Cyclobutane-containing peptides: Evaluation as novel metallocarboxypeptidase inhibitors and modelling of their mode of action

Daniel Fernández, Elisabeth Torres, Francesc Avilés, Rosa M. Ortuño, Josep Vendrell

Bioorganic & Medicinal Chemistry · 2009 · 45 citations · 26 references

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References

26

Relationship between the inhibition constant (KI) and the concentration of inhibitor which causes 50 per cent inhibition (I50) of an enzymatic reaction

Yung-Chi Cheng, William H. Prusoff · Biochemical Pharmacology · 1973 · 12.9K citations

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The Outstanding Biological Stability ofβ- andγ-Peptides toward Proteolytic Enzymes: An In Vitro Investigation with Fifteen Peptidases

Jens Frackenpohl, Per I. Arvidsson, Jürg V. Schreiber et al. · ChemBioChem · 2001 · 406 citations

, , +17

Carboxypeptidase E mediates palmitate-induced β-cell ER stress and apoptosis

Kristin D. Jeffrey, Emilyn U. Alejandro, Dan S. Luciani et al. · Proceedings of the National Academy of Sciences · 2008 · 149 citations · Full text

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Nnal‐like proteins are active metallocarboxypeptidases of a new and diverse M14 subfamily

Mónica Rodríguez de la Vega, Rafael G. Sevilla, Antonio Hermoso et al. · The FASEB Journal · 2007 · 113 citations

, , +14

Serum levels of procarboxypeptidase B and its activation peptide in patients with acute pancreatitis and non-pancreatic diseases

Christophe Müller, Stefan Appelros, Waldemar Uhl et al. · Gut · 2002 · 62 citations · Full text

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