In vitro and in vivo effects of kelatorphan on enkephalin metabolism in rodent brain

PHARMACOLOGICAL EFFECTS PRODUCED BY INTRACEREBRAL INJECTION OF DRUGS IN THE CONSCIOUS MOUSE

Thomas J. Haley, WF McCormick · British Journal of Pharmacology and Chemotherapy · 1957 · 1.5K citations · Full text

Local Pharmacology, Pharmacotherapy, Experimental Pharmacology +16

Proteinases in mammalian cells and tissues

Michael Kerr · Biochemical Education · 1978 · 922 citations

Protein Expression, Cellular Enzymology, Biochemistry +8

Design of potent competitive inhibitors of angiotensin-converting enzyme. Carboxyalkanoyl and mercaptoalkanoyl amino acids

David W. Cushman, H.S. Cheung, Emily F. Sabo et al. · Biochemistry · 1977 · 900 citations

Cardiovascular Pharmacology, Altmetric Attention Score, Pharmacotherapy +17

The enkephalinase inhibitor thiorphan shows antinociceptive activity in mice

B P Roques, M C Fournié-Zaluski, E. Soroca et al. · Nature · 1980 · 707 citations

Inflammation, Molecular Pharmacology, Health Sciences +10

High-affinity enkephalin-degrading peptidase in brain is increased after morphine

Bernard Malfroy, Jean-Paul Swerts, Anne Guyon et al. · Nature · 1978 · 650 citations

Molecular Pharmacology, Molecular Neuroscience, Medicine +8