Concepedia

Design, synthesis, and biological evaluation of quinazoline derivatives as α-glucosidase inhibitors

Venkateshwarlu Gurram, Ramesh Garlapati, T. Chiranjeevi, Nagaraju Madala, Kumara Swamy Kasani, Pavan Kumar Machiraju, Raju Doddapalla, Uma Addepally, Rambabu Gundla, Balaram Patro,

Medicinal Chemistry Research · 2014 · 29 citations · 23 references

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References

23

Glide:  A New Approach for Rapid, Accurate Docking and Scoring. 1. Method and Assessment of Docking Accuracy

Richard A. Friesner, Jay L. Banks, Robert B. Murphy et al. · Journal of Medicinal Chemistry · 2004 · 9.9K citations

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Empirical scoring functions: I. The development of a fast empirical scoring function to estimate the binding affinity of ligands in receptor complexes

Matthew Eldridge, Christopher W. Murray, T.R. Auton et al. · Journal of Computer-Aided Molecular Design · 1997 · 1.7K citations

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Molecular Shape Diversity of Combinatorial Libraries:  A Prerequisite for Broad Bioactivity

Wolfgang Sauer, Matthias Schwarz · Journal of Chemical Information and Computer Sciences · 2003 · 496 citations

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Quinazolinone Derivatives as Orally Available Ghrelin Receptor Antagonists for the Treatment of Diabetes and Obesity

Joachim Rudolph, William P. Esler, Stephen O’Connor et al. · Journal of Medicinal Chemistry · 2007 · 157 citations · Full text

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Discovery of novel α-glucosidase inhibitors based on the virtual screening with the homology-modeled protein structure

Hwangseo Park, Kyo Yeol Hwang, Kyung Hwan Oh et al. · Bioorganic & Medicinal Chemistry · 2007 · 124 citations

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