The G protein-coupled receptor GPR30 mediates the proliferative and invasive effects induced by hydroxytamoxifen in endometrial cancer cells

A Transmembrane Intracellular Estrogen Receptor Mediates Rapid Cell Signaling

Chetana M. Revankar, Daniel F. Cimino, Larry A. Sklar et al. · Science · 2005 · 2.3K citations

Life Sciences, Biochemistry, Cell Biology +10

Identity of an Estrogen Membrane Receptor Coupled to a G Protein in Human Breast Cancer Cells

Peter Thomas, Yefei Pang, Edward J. Filardo et al. · Endocrinology · 2004 · 1.4K citations · Full text

Life Sciences, Endocrinology, Molecular Biology +17

Estrogen-Induced Activation of Erk-1 and Erk-2 Requires the G Protein-Coupled Receptor Homolog, GPR30, and Occurs via Trans-Activation of the Epidermal Growth Factor Receptor through Release of HB-EGF

Edward J. Filardo, Jeffrey A. Quinn, Kirby I. Bland et al. · Molecular Endocrinology · 2000 · 1.3K citations · Full text

Life Sciences, Biochemistry, Molecular Biology +17

Estrogen Action Via the G Protein-Coupled Receptor, GPR30: Stimulation of Adenylyl Cyclase and cAMP-Mediated Attenuation of the Epidermal Growth Factor Receptor-to-MAPK Signaling Axis

Edward J. Filardo, Jeffrey A. Quinn, A. Raymond Frackelton et al. · Molecular Endocrinology · 2002 · 854 citations · Full text

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Coactivator and Corepressor Regulation of the Agonist/Antagonist Activity of the Mixed Antiestrogen, 4-Hydroxytamoxifen

C. Smith, Zafar Nawaz, Bert W. O’Malley · Molecular Endocrinology · 1997 · 643 citations

Life Sciences, Endocrinology, Pharmacology +17