Concepedia

Indole- and benzothiophene-based histamine H3 antagonists

Alejandro Santillán, Kelly J. McClure, Brett D. Allison, Brian Lord, Jamin D. Boggs, Kirsten L. Morton, Anita Everson, Diane Nepomuceno, Michael A. Letavic, Alice Lee-Dutra,

Bioorganic & Medicinal Chemistry Letters · 2010 · 12 citations · 14 references

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14

Auto-inhibition of brain histamine release mediated by a novel class (H3) of histamine receptor

Jean‐Michel Arrang, M. Garbarg, Jean‐Charles Schwartz · Nature · 1983 · 1.6K citations

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Autoinhibition of histamine synthesis mediated by presynaptic H3-receptors

JM Arrang, M. Garbarg, Schwartz Jc · Neuroscience · 1987 · 267 citations

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Validation of a [3H]Astemizole Binding Assay in HEK293 Cells Expressing HERG K+ Channels

Peter Chiu, Karen F. Marcoe, Sidney E. Bounds et al. · Journal of Pharmacological Sciences · 2004 · 134 citations · Full text

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[3H]Dofetilide binding to HERG transfected membranes: a potential high throughput preclinical screen

Keith Finlayson, L Turnbull, Craig T. January et al. · European Journal of Pharmacology · 2001 · 131 citations

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4-(2-[2-(2(<i>R</i>)-Methylpyrrolidin-1-yl)ethyl]benzofuran-5-yl)benzonitrile and Related 2-Aminoethylbenzofuran H<sub>3</sub> Receptor Antagonists Potently Enhance Cognition and Attention

Marlon Cowart, Ramin Faghih, Michael P. Curtis et al. · Journal of Medicinal Chemistry · 2004 · 122 citations · Full text

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