Concepedia

Synthesis and in vitro EGFR (ErbB1) tyrosine kinase inhibitory activity of 4-N-substituted 6-aryl-7H-pyrrolo[2,3-d]pyrimidine-4-amines

Svein Jacob Kaspersen, Christopher Sørum, Veronica Willassen, Erik Fuglseth, Eli Kjøbli, Geir Bjørkøy, Eirik Sundby, Bård Helge Hoff

European Journal of Medicinal Chemistry · 2011 · 37 citations · 22 references

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22

AutoDock Vina: Improving the speed and accuracy of docking with a new scoring function, efficient optimization, and multithreading

Oleg Trott, Arthur J. Olson · Journal of Computational Chemistry · 2009 · 37.1K citations · Full text

, , +17

Python: a programming language for software integration and development.

M F Sanner · PubMed · 1999 · 3.1K citations

, , +11

Structures of Lung Cancer-Derived EGFR Mutants and Inhibitor Complexes: Mechanism of Activation and Insights into Differential Inhibitor Sensitivity

Cai‐Hong Yun, Titus J. Boggon, Yiqun Li et al. · Cancer Cell · 2007 · 1.2K citations · Full text

, , +15

Thousands of chemical starting points for antimalarial lead identification

Francisco‐Javier Gamo, Laura M. Sanz, Jaume Vidal et al. · Nature · 2010 · 1K citations

, , +12

The Selective Reaction of Aryl Halides with KOH:  Synthesis of Phenols, Aromatic Ethers, and Benzofurans

Kevin W. Anderson, Takashi Ikawa, Rachel E. Tundel et al. · Journal of the American Chemical Society · 2006 · 461 citations

, , +10