Nociceptin/Orphanin FQ Receptor Activation Attenuates Antinociception Induced by Mixed Nociceptin/Orphanin FQ/μ-Opioid Receptor Agonists

Relationship between the inhibition constant (KI) and the concentration of inhibitor which causes 50 per cent inhibition (I50) of an enzymatic reaction

Yung-Chi Cheng, William H. Prusoff · Biochemical Pharmacology · 1973 · 12.9K citations

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Isolation and structure of the endogenous agonist of opioid receptor-like ORL1 receptor

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Orphanin FQ: A Neuropeptide That Activates an Opioidlike G Protein-Coupled Receptor

Rainer K. Reinscheid, Hans‐Peter Nothacker, Anne Bourson et al. · Science · 1995 · 1.8K citations

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Human Pharmacology and Abuse Potential of the Analgesic Buprenorphine

Donald R. Jasinski · Archives of General Psychiatry · 1978 · 787 citations

Medicine, Pharmacology, Pharmacotherapy +11

AGONIST AND ANTAGONIST PROPERTIES OF BUPRENORPHINE, A NEW ANTINOCICEPTIVE AGENT

A. Cowan, John W. Lewis, Ian R. Macfarlane · British Journal of Pharmacology · 1977 · 528 citations · Full text

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