Concepedia

Synthesis of C-cinnamoyl glycosides and their inhibitory activity against mammalian carbonic anhydrases

Leonardo E. Riafrecha, Oscar M. Rodríguez, Daniela Vullo, Claudiu T. Supuran, Pedro A. Colinas

Bioorganic & Medicinal Chemistry · 2012 · 36 citations · 25 references

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References

25

Relationship between the inhibition constant (KI) and the concentration of inhibitor which causes 50 per cent inhibition (I50) of an enzymatic reaction

Yung-Chi Cheng, William H. Prusoff · Biochemical Pharmacology · 1973 · 12.9K citations

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Fast Calculation of Molecular Polar Surface Area as a Sum of Fragment-Based Contributions and Its Application to the Prediction of Drug Transport Properties

Peter Ertl, Bernhard Rohde, Paul M. Selzer · Journal of Medicinal Chemistry · 2000 · 3K citations

, , +15

The Carbon Dioxide Hydration Activity of Carbonic Anhydrase

Raja G. Khalifah · Journal of Biological Chemistry · 1971 · 1.9K citations · Full text

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Carbonic anhydrase inhibitors

Claudiu T. Supuran, Andrea Scozzafava, Angela Casini · Medicinal Research Reviews · 2002 · 1.4K citations

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Non-Zinc Mediated Inhibition of Carbonic Anhydrases: Coumarins Are a New Class of Suicide Inhibitors

Alfonso Maresca, Claudia Temperini, Hoan Vu et al. · Journal of the American Chemical Society · 2009 · 512 citations · Full text

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