Bioorganic & Medicinal Chemistry Letters · 2000 · 12 citations · 6 references
PharmacyMedicinal ChemistryPharmacologyDrug DesignDrug DiscoveryLead OptimizationCovalent Inhibitor DesignDe Novo Drug DesignEnzyme DesignEnzyme InhibitionLead Compound DesignPotency OptimizationCysteine-targeted InhibitorsEnzyme Inhibitor SynthesisThiol Chemistry
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A novel potent vasoconstrictor peptide produced by vascular endothelial cells
Masashi Yanagisawa, Hiroki Kurihara, Sadao Kimura et al. · Nature · 1988 · 10.8K citations · Full text