Substance P (NK-1 receptor) antagonists: In vivo and in vitro activities in rats and guinea pigs

A Potent Nonpeptide Antagonist of the Substance P (NK ₁ ) Receptor

R. Michael Snider, Jay W. Constantine, John Lowe et al. · Science · 1991 · 864 citations

Medicine, Medicinal Chemistry, Pharmacology +14

A potent and selective non-peptide antagonist of the neurokinin a (NK2) receptor

Xavier Emonds‐Alt, P. Vilain, P. Goulaouic et al. · Life Sciences · 1992 · 437 citations

Medicine, Neuroscience, Pharmacology +5

Investigation into species variants in tachykinin NK₁ receptors by use of the non‐peptide antagonist, CP‐96,345

I.J.M. Beresford, P.J. Birch, R.M. Hagan et al. · British Journal of Pharmacology · 1991 · 220 citations · Full text

Medicine, Pharmacology, Comparative Pharmacology +13

Neurokinin A (NK2) receptor revisited with SR 48968, a potent non-peptide antagonist

Charles Advenier, N. Rouissi, Quang T. Nguyen et al. · Biochemical and Biophysical Research Communications · 1992 · 168 citations

Medicine, Neuroscience, Pharmacology +7

Species differences in affinities of non-peptide antagonists for substance p receptors

Bruce D. Gitter, Diane C. Waters, Robert F. Bruns et al. · European Journal of Pharmacology · 1991 · 163 citations

Medicine, Pharmacology, General Pharmacology +15