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Selective CB2 agonists with anti-pruritic activity: Discovery of potent and orally available bicyclic 2-pyridones

Ken‐ichi Kusakabe, Yasuyoshi Iso, Yukio Tada, Masahiro Sakagami, Yasuhide Morioka, Nobuo Chomei, Satomi Shinonome, Keiko Kawamoto, Hideyuki Takenaka, Kiyoshi Yasui,

Bioorganic & Medicinal Chemistry · 2013 · 18 citations · 23 references

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23

Crystal structure of the β2 adrenergic receptor–Gs protein complex

Søren G. F. Rasmussen, Brian T. DeVree, Yaozhong Zou et al. · Nature · 2011 · 3.1K citations · Full text

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Evaluation of binding in a transfected cell line expressing a peripheral cannabinoid receptor (CB2): identification of cannabinoid receptor subtype selective ligands.

Vincent M. Showalter, David M. Compton, BR Martin et al. · Journal of Pharmacology and Experimental Therapeutics · 1996 · 572 citations

, , +14

HU-308: A specific agonist for CB <sub>2</sub> , a peripheral cannabinoid receptor

L Hanŭs, Aviva Breuer, Susanna Tchilibon et al. · Proceedings of the National Academy of Sciences · 1999 · 568 citations · Full text

, , +17

Cannabinoid structure-activity relationships: correlation of receptor binding and in vivo activities.

David M. Compton, Kenner C. Rice, Barbara Costa et al. · Journal of Pharmacology and Experimental Therapeutics · 1993 · 464 citations · Full text

, , +17

CB2 cannabinoid receptor-mediated peripheral antinociception

Philip T. Malan, Mohab Ibrahim, Hongfeng Deng et al. · Pain · 2001 · 389 citations

, , +14