Concepedia
Bioorganic & Medicinal Chemistry · 2004 · 105 citations · 24 references
Molecular PharmacologyFunctional SelectivityMedicineDrug DiscoveryMechanism Of ActionPharmacological AgentVitro BindingDopaminePharmacologyN-phenyl Piperazine AnalogsBiomolecular Engineering
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Relationship between the inhibition constant (KI) and the concentration of inhibitor which causes 50 per cent inhibition (I50) of an enzymatic reaction
Yung-Chi Cheng, William H. Prusoff · Biochemical Pharmacology · 1973 · 12.8K citations
Cent Inhibition, Inhibitory Activity, Biochemistry +8
A RADIOISOTOPIC METHOD FOR MEASURING THE FORMATION OF ADENOSINE 3′,5′‐CYCLIC MONOPHOSPHATE IN INCUBATED SLICES OF BRAIN
Hirotoshi Shimizu, John W. Daly, Cyrus R. Creveling · Journal of Neurochemistry · 1969 · 468 citations
Experimental Pharmacology, Social Sciences, Adenosine 3′,5′‐Cyclic +17
Distribution of Dopamine D3 Receptor Expressing Neurons in the Human Forebrain Comparison with D2 Receptor Expressing Neurons
Eugenia V. Gurevich · Neuropsychopharmacology · 1999 · 431 citations
Human Forebrain Comparison, Neuroanatomy, Physiology +11
Relationship between lipophilicity and brain extraction of C-11-labeled radiopharmaceuticals.
Douglas D. Dischino, Michael J. Welch, Michael R. Kilbourn et al. · PubMed · 1983 · 286 citations
Engineering, Cerebral Vascular Regulation, Blood Flow +19
Mesolimbic Dopamine D3 Receptors and Use of Antipsychotics in Patients With Schizophrenia
Eugenia V. Gurevich · Archives of General Psychiatry · 1997 · 247 citations