Application of copper(I)-catalysed azide/alkyne cycloaddition (CuAAC) ‘click chemistry’ in carbohydrate drug and neoglycopolymer synthesis

Click Chemistry: Diverse Chemical Function from a Few Good Reactions

Hartmuth C. Kolb, M. G. Finn, K. Barry Sharpless · Angewandte Chemie International Edition · 2001 · 12.9K citations

Combinatorial Chemistry, Click Chemistry Status, Engineering +17

A Stepwise Huisgen Cycloaddition Process: Copper(I)-Catalyzed Regioselective “Ligation” of Azides and Terminal Alkynes

Vsevolod V. Rostovtsev, Luke G. Green, Valery V. Fokin et al. · Angewandte Chemie International Edition · 2002 · 11.4K citations

Terminal Alkynes, Chemical Engineering, Novel Organocatalysts +12

Click Chemistry: Diverse Chemical Function from a Few Good Reactions

Hartmuth C. Kolb, M. G. Finn, K. Barry Sharpless · Angewandte Chemie International Edition · 2001 · 9.3K citations · Full text

Peptidotriazoles on Solid Phase:  [1,2,3]-Triazoles by Regiospecific Copper(I)-Catalyzed 1,3-Dipolar Cycloadditions of Terminal Alkynes to Azides

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Terminal Alkynes, Novel Organocatalysts, Solid Phase +15

The Properties of Known Drugs. 1. Molecular Frameworks

Guy W. Bemis, Mark A. Murcko · Journal of Medicinal Chemistry · 1996 · 2.3K citations

Molecular Docking, Molecular Pharmacology, Medicinal Chemistry +15