Synthesis of 3-aminopyrrolidines and piperidines from endocyclic enamine derivatives

A three-component coupling protocol for the synthesis of substituted hexahydropyrrolo[3,2-c]quinolines

Robert A. Batey, Paul D. Simoncic, Denny Lin et al. · Chemical Communications · 1999 · 93 citations

Natural Sciences, Chemistry, Medicinal Chemistry +8

Azaglycosylation of complex stannyl alkoxides with glycal-derived iodo sulfonamides: a straightforward synthesis of sialyl-Lewis X antigen and other oligosaccharide domains

Samuel J. Danishefsky, Koshi Koseki, David A. Griffith et al. · Journal of the American Chemical Society · 1992 · 83 citations

Life Sciences, Biochemistry, Chemistry +14

Phenylaziridine as a 1,3-dipole. Application to the synthesis of functionalized pyrrolidines

Ioana Ungureanu, Cristian Bologa, Saïd Chayer et al. · Tetrahedron Letters · 1999 · 47 citations

Natural Sciences, Chemistry, Medicinal Chemistry +4

Stereoselective synthesis of (+)-CP-99,994: A substance P non-peptide antagonist

S. Chandrasekhar, Pradyumna K. Mohanty · Tetrahedron Letters · 1999 · 37 citations

Pharmacy, Medicinal Chemistry, Pharmacology +6

First asymmetric synthesis of (2R, 3R)-3-amino-1-benzyl-2-methyl-pyrrolidine via a highly diastereoselective reductive alkylation

Pei‐Qiang Huang, Si Li Wang, Hong Zheng et al. · Tetrahedron Letters · 1997 · 37 citations

Natural Sciences, Chemistry, Medicinal Chemistry +8