Binding characteristics of γ-hydroxybutyric acid as a weak but selective GABAB receptor agonist

Relationship between the inhibition constant (KI) and the concentration of inhibitor which causes 50 per cent inhibition (I50) of an enzymatic reaction

Yung-Chi Cheng, William H. Prusoff · Biochemical Pharmacology · 1973 · 12.9K citations

Life Sciences, Biochemistry, Chemical Kinetics +14

3H-baclofen and 3H-GABA bind to bicuculline-insensitive GABAB sites in rat brain

David R. Hill, Norman G. Bowery · Nature · 1981 · 1K citations

Life Sciences, Neuroscience, Pharmacology +16

GABAA and GABAB receptor site distribution in the rat central nervous system

Norman G. Bowery, Alan L. Hudson, Geraint Price · Neuroscience · 1987 · 862 citations

Life Sciences, Neurobiology, Neuroscience +14

High affinity binding site for γ-hydroxybutyric acid in rat brain

Jesús Bénavidès, J.F. Rumigny, Jean‐Jacques Bourguignon et al. · Life Sciences · 1982 · 207 citations

Life Sciences, Neurobiology, Neuroscience +12

Evidence for GABAB-mediated mechanisms in experimental generalized absence seizures

O. Carter Snead · European Journal of Pharmacology · 1992 · 172 citations

Life Sciences, Neurobiology, Neuroscience +14