Concepedia

Synthesis and activity of pyrrolidinyl- and thiazolidinyl-dipeptide derivatives as inhibitors of the Tc80 prolyl oligopeptidase from Trypanosoma cruzi

Roger Joyeau, Chanfi Maoulida, C. Guillet, François Frappier, Antônio R. L. Teixeira, Joseph Schrével, Jaime M. Santana, Philippe Grellier

European Journal of Medicinal Chemistry · 2000 · 31 citations · 36 references

DOI

Concepts

References

36

N-methoxy-n-methylamides as effective acylating agents

Steven Nahm, Steven M. Weinreb · Tetrahedron Letters · 1981 · 1.8K citations

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Proteolytic enzymes; a practical approach

Comparative Biochemistry and Physiology Part A Physiology · 1991 · 762 citations

, , +14

A linear equation that describes the steady-state kinetics of enzymes and subcellular particles interacting with tightly bound inhibitors

Peter J. F. Henderson · Biochemical Journal · 1972 · 524 citations · Full text

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Vinyl Sulfones as Mechanism-Based Cysteine Protease Inhibitors

James T. Palmer, David Rasnick, Jeffrey L. Klaus et al. · Journal of Medicinal Chemistry · 1995 · 506 citations · Full text

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Prolyl Oligopeptidase

Vilmos Fülöp, Zsolt Böcskei, László Polgár · Cell · 1998 · 494 citations · Full text