Concepedia

Tetrahydroisoquinoline-3-carboxylate based matrix-metalloproteinase inhibitors: design, synthesis and structure–activity relationship

Hans Matter, Manfred Schudok, Wilfried Schwab, Werner Thorwart, Denis Barbier, Günter Billen, Burkhard Haase, Bernhard Neises, Klaus-Ulrich Weithmann, Theo Wollmann

Bioorganic & Medicinal Chemistry · 2002 · 56 citations · 33 references

DOI

Concepts

References

33

The protein data bank: A computer-based archival file for macromolecular structures

F. C. Bernstein, Thomas F. Koetzle, G. J. B. Williams et al. · Journal of Molecular Biology · 1977 · 8.6K citations

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On the size of the active site in proteases. I. Papain

Israël Schechter, Arieh Berger · Biochemical and Biophysical Research Communications · 1967 · 5.2K citations

, , +9

Iterative partial equalization of orbital electronegativity—a rapid access to atomic charges

Johann Gasteiger, Mario Marsili · Tetrahedron · 1980 · 4.1K citations

, , +10

Comparative molecular field analysis (CoMFA). 1. Effect of shape on binding of steroids to carrier proteins

Richard D. Cramer, David E. Patterson, Jeffrey D. Bunce · Journal of the American Chemical Society · 1988 · 3.9K citations

, , +14

Matrix metalloproteinases and their inhibitors in connective tissue remodeling

J. Frederick Woessner · The FASEB Journal · 1991 · 3.3K citations · Full text

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