The nature of inhibition of steroid sulphatase activity by tibolone and its metabolites

Estrone sulfamates: potent inhibitors of estrone sulfatase with therapeutic potential

Nicola M. Howarth, Atul Purohit, Michael Reed et al. · Journal of Medicinal Chemistry · 1994 · 218 citations · Full text

Medicine, Medicinal Chemistry, Pharmacology +11

THE RELATIONSHIP BETWEEN 17β‐HYDROXYSTEROID DEHYDROGENASE ACTIVITY AND OESTROGEN CONCENTRATIONS IN HUMAN BREAST TUMOURS AND IN NORMAL BREAST TISSUE

Rosemary C. Bonney, Michael Reed, Kathryn Davidson et al. · Clinical Endocrinology · 1983 · 187 citations

Life Sciences, Biochemistry, Oncology +17

Inactivation of Steroid Sulfatase by an Active Site-Directed Inhibitor, Estrone-3-O-Sulfamate

Atul Purohit, Gary J. Williams, Nicola M. Howarth et al. · Biochemistry · 1995 · 170 citations

Life Sciences, Biochemistry, Pharmacology +13

Systemic Distribution of Steroid Sulfatase and Estrogen Sulfotransferase in Human Adult and Fetal Tissues

Yasuhiro Miki, Taisuke Nakata, Takashi Suzuki et al. · The Journal of Clinical Endocrinology & Metabolism · 2002 · 169 citations · Full text

Life Sciences, Biochemistry, Endocrinology +16

In vitro evaluation of estrogenic, estrogen antagonistic and progestagenic effects of a steroidal drug (Org OD-14) and its metabolites on human endometrium

Leszek Markiewicz, Erlio Gurpide · Journal of Steroid Biochemistry · 1990 · 113 citations

Medicine, Endocrinology, Pharmacology +12