Concepedia

Nonpeptide endothelin antagonists: from lower affinity pyrazol-5-ols to higher affinity pyrazole-5-carboxylic acids

Jidong Zhang, Stanislas Didierlaurent, Michel Fortin, Dominique Lefrançois, Eric Uridat, Jean Paul Vevert

Bioorganic & Medicinal Chemistry Letters · 2000 · 24 citations · 28 references

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References

28

A novel potent vasoconstrictor peptide produced by vascular endothelial cells

Masashi Yanagisawa, Hiroki Kurihara, Sadao Kimura et al. · Nature · 1988 · 10.8K citations · Full text

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Comprehensive organic chemistry

D. H. R. BARTON, W. David Ollis · Tetrahedron Letters · 1978 · 2.8K citations

Cloning and expression of a cDNA encoding an endothelin receptor

Hiroshi Arai, Seiji Hori, Ichiro Aramori et al. · Nature · 1990 · 2.6K citations

, , +7

Cloning of a cDNA encoding a non-isopeptide-selective subtype of the endothelin receptor

Takeshi Sakurai, Masashi Yanagisawa, Yoh Takuwat et al. · Nature · 1990 · 2.4K citations · Full text

, , +8

Biological profiles of highly potent novel endothelin antagonists selective for the ETA receptor

Masaki Ihara, Kazuhito Noguchi, Toshihiko Saeki et al. · Life Sciences · 1992 · 877 citations

, , +7