Journal of the Chemical Society Perkin Transactions 1 · 1995 · 32 citations · 24 references
Natural SciencesChemistryMedicinal ChemistryCancer PharmacologyDrug DiscoveryOrganic ChemistryHeterocyclic ChemistryStereochemical OptimizationStereoselective C-h FunctionalizationStereoselective Reaction DesignStereoselective SynthesisStereoselectivityStereoselectivity ControlStereoselectivity In Addition ReactionsStereoselectivity OptimizationStereospecific Reaction Design
The C-2 methylated 2S,3R and 2R,3S side chains of docetaxel have been enantioselectively prepared and esterified with protected 10-deacetylbaccatin III to provide novel analogues of docetaxel.
24
K. C. Nicolaou, Zhen Yang, Jimei Liu et al. · Nature · 1994 · 1.1K citations
The Alkaloids, Chemistry and Pharmacology
European Journal of Medicinal Chemistry · 1992 · 916 citations