N-Benzylgalactonoamidines as potent β-galactosidase inhibitors

1-Aza Sugars, Apparent Transition State Analogues of Equatorial Glycoside Formation/Cleavage

Mikael Bols · Accounts of Chemical Research · 1998 · 264 citations

Pharmacy, Biochemistry, Chemistry +9

Synthesis and Evaluation of Homoaza Sugars as Glycosidase Inhibitors

Chi‐Huey Wong, Louis Provencher, John A. Porco et al. · The Journal of Organic Chemistry · 1995 · 146 citations

Life Sciences, Biochemistry, Medicinal Chemistry +9

An ab initio study (6-31G*) of transition states in glycoside hydrolysis based on axial and equatorial 2-methoxytetrahydropyrans

C. Webster Andrews, Bert Fraser‐Reid, J. Phillip Bowen · Journal of the American Chemical Society · 1991 · 104 citations

Life Sciences, Biochemistry, Chemistry +13

Potent, broad-spectrum inhibition of glycosidases by an amidine derivative of D-glucose

Michael K. Tong, George Papandreou, Bruce Ganem · Journal of the American Chemical Society · 1990 · 90 citations

Life Sciences, Biochemistry, Pharmacology +9

Configurationally selective transition state analogue inhibitors of glycosidases. A study with nojiritetrazoles, a new class of glycosidase inhibitors

Philipp Ermert, Andrea Vasella, Martin Weber et al. · Carbohydrate Research · 1993 · 72 citations

Life Sciences, Biochemistry, Medicinal Chemistry +13