Potent inhibition of protein-tyrosine phosphatese-1B using the phosphotyrosyl mimetic fluoro-O-malonyl tyrosine (FOMT)

Potent Inhibition of Insulin Receptor Dephosphorylation by a Hexamer Peptide Containing the Phosphotyrosyl Mimetic F2Pmp

Terrence R. Burke, Hemanta K. Kole, Peter P. Roller · Biochemical and Biophysical Research Communications · 1994 · 208 citations

Life Sciences, Biochemistry, Endocrinology +16

Protein Tyrosine Phosphatase Substrate Specificity: Size and Phosphotyrosine Positioning Requirements in Peptide Substrates

Zhong Yin Zhang, Derek Maclean, Dennis J. McNamara et al. · Biochemistry · 1994 · 172 citations

Life Sciences, Biochemistry, Molecular Biology +14

Preparation of fluoro- and hydroxy-4-(phosphonomethyl)-D,L-phenylalanine suitably protected for solid-phase synthesis of peptides containing hydrolytically stable analogs of O-phosphotyrosine

Terrence R. Burke, Mark S. Smyth, Motoyoshi Nomizu et al. · The Journal of Organic Chemistry · 1993 · 162 citations

Natural Sciences, Biochemistry, Chemistry +10

4‘-<i>O</i>-[2-(2-Fluoromalonyl)]-<scp>l</scp>-tyrosine:  A Phosphotyrosyl Mimic for the Preparation of Signal Transduction Inhibitory Peptides

Bin Ye, Miki Akamatsu, Harry Ford et al. · Journal of Medicinal Chemistry · 1996 · 96 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +17

Synthesis of new amino acids mimicking sulfated and phosphorylated tyrosine residues

I. Marseigne, B.P. Roques · The Journal of Organic Chemistry · 1988 · 81 citations

Life Sciences, Biochemistry, Chemistry +13