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Methylation of imidazoline related compounds leads to loss of α2-adrenoceptor affinity. Synthesis and biological evaluation of selective I1 imidazoline receptor ligands

Stéphan Schann, Hugues Greney, Vincent Gasparik, Monique Dontenwill, Carla Rascente, Gabriel Lacroix, Laurent Monassier, Véronique Bruban, Josiane Feldman, Jean‐Daniel Ehrhardt,

Bioorganic & Medicinal Chemistry · 2012 · 13 citations · 28 references

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28

Agmatine: an Endogenous Clonidine-Displacing Substance in the Brain

Gen Li, S. Regunathan, Colin J. Barrow et al. · Science · 1994 · 751 citations

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Moxonidine, a centrally acting antihypertensive agent, is a selective ligand for I1-imidazoline sites.

Paul Ernsberger, T. H. Damon, LYNETTE M. GRAFF et al. · Journal of Pharmacology and Experimental Therapeutics · 1993 · 245 citations

, , +17

Localization of I2-Imidazoline Binding Sites on Monoamine Oxidases

Frédérique Tesson, Isabelle Limon, Philippe Urban et al. · Journal of Biological Chemistry · 1995 · 174 citations · Full text

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Isolation and partial purification of a clonidine‐displacing endogenous brain substance

Daphné Atlas, Yigal Burstein · European Journal of Biochemistry · 1984 · 148 citations · Full text

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Actions of α2 adrenoceptor ligands at α2A and 5-HT1A receptors: the antagonist, atipamezole, and the agonist, dexmedetomidine, are highly selective for α2A adrenoceptors

Adrian Newman‐Tancredi, Jean‐Paul Nicolas, Valérie Audinot et al. · Naunyn-Schmiedeberg s Archives of Pharmacology · 1998 · 119 citations

, , +11