Concepedia

Synthesis and evaluation of a γ-lactam as a highly selective EP2 and EP4 receptor agonist

Yufang Xiao, Gian Luca Araldi, Zhong Zhao, Adulla Reddy, Srinivasa Karra, Nadia Brügger, David Fischer, Elizabeth E. Palmer, Bagna Bao, Sean D. McKenna

Bioorganic & Medicinal Chemistry Letters · 2007 · 14 citations · 10 references

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10

A stable and easily prepared catalyst for the enantioselective reduction of ketones. Applications to multistep syntheses

E. J. Corey, Raman K. Bakshi, Saizo Shibata et al. · Journal of the American Chemical Society · 1987 · 864 citations

, , +15

Prostaglandin E2 Suppresses Chemokine Production in Human Macrophages through the EP4 Receptor

Kiyoshi Takayama, Guillermo García‐Cardeña, Galina K. Sukhova et al. · Journal of Biological Chemistry · 2002 · 338 citations · Full text

, , +17

Molecular cloning and characterization of the four rat prostaglandin E2 prostanoid receptor subtypes

Yves Boie, Rino Stocco, Nicole Sawyer et al. · European Journal of Pharmacology · 1997 · 299 citations

, , +7

LY171883, 1-less than 2-hydroxy-3-propyl-4-less than 4-(1H-tetrazol-5-yl) butoxy greater than phenyl greater than ethanone, an orally active leukotriene D4 antagonist.

J H Fleisch, Lynn E. Rinkema, Klaus D. Haisch et al. · Journal of Pharmacology and Experimental Therapeutics · 1985 · 163 citations

, , +10

Characterization of prostanoid relaxant/inhibitory receptors (ψ) using a highly selective agonist, TR4979

Phillip J. Gardiner · British Journal of Pharmacology · 1986 · 147 citations · Full text

, , +13