Asymmetric synthesis of α-amino acids from carbohydrates as chiral templates

Asymmetric glycine enolate aldol reactions: synthesis of cyclosporin's unusual amino acid, MeBmt

David A. Evans, Ann E. Weber · Journal of the American Chemical Society · 1986 · 343 citations

Natural Sciences, Biochemistry, Medicinal Chemistry +8

Stereoselective Syntheses of Building Blocks with Three Consecutive Stereogenic Centers: Important Precursors of Polyketide Natural Products [New Synthetic Methods (68)]

Reinhard W. Hoffmann · Angewandte Chemie International Edition in English · 1987 · 218 citations

Pharmacy, Chemistry, Carbohydrate Chemistry +10

Asymmetric synthesis on carbohydrate templates: stereoselective Ugi-synthesis of .alpha.-amino acid derivatives

Horst Kunz, Waldemar Pfrengle · Journal of the American Chemical Society · 1988 · 168 citations

Natural Sciences, Biochemistry, Chemistry +11

Synthesis of cyclosporine. Total syntheses of ‘cyclosporin A’ and ‘cyclosporin H’, two fungal metabolites isolated from the species <i>Tolypocladium inflatum</i> G<scp>AMS</scp>

Roland M. Wenger · Helvetica Chimica Acta · 1984 · 159 citations

Pharmacy, Chemistry, Medicinal Chemistry +15

Formation of convenient chiral intermediates from carbohydrates and their use in synthesis

Thomas D. Inch · Tetrahedron · 1984 · 152 citations

Pharmacy, Biochemistry, Chemistry +12