Concepedia

Studies on the chemistry of thienoanellated O,N- and S,N-containing heterocycles. Part 30: Synthesis and pharmacological properties of thieno[2,3-b][1,4]thiazines with potential vasopressin receptor antagonistic activity

Maria E. Galanski, Thomas Erker, Norbert Handler, Rosa Lemmens‐Gruber, M. Kamyar, Christian Studenik

Bioorganic & Medicinal Chemistry · 2005 · 17 citations · 18 references

DOI

Concepts

References

18

Characterization of a novel aquaretic agent, OPC‐31260, as an orally effective, nonpeptide vasopressin V<sub>2</sub> receptor antagonist

Yoshitaka Yamamura, Hidenori Ogawa, Hiroshi Yamashita et al. · British Journal of Pharmacology · 1992 · 347 citations · Full text

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OPC-21268, an Orally Effective, Nonpeptide Vasopressin V1 Receptor Antagonist

Yoshitaka Yamamura, Hidenori Ogawa, Tomihiko Chihara et al. · Science · 1991 · 272 citations

, , +17

Characterization of SR 121463A, a highly potent and selective, orally active vasopressin V2 receptor antagonist.

C. Serradeil‐Le Gal, C Lacour, G Valette et al. · Journal of Clinical Investigation · 1996 · 249 citations · Full text

, , +11

Coronary vasoconstriction induced by vasopressin. Production of myocardial ischemia in dogs by constriction of nondiseased small vessels.

Mary F. Maturi, Staci Martin, David R. Markle et al. · Circulation · 1991 · 89 citations

, , +14

Orally Active, Nonpeptide Vasopressin V<sub>2</sub> Receptor Antagonists:  A Novel Series of 1-[4-(Benzoylamino)benzoyl]-2,3,4,5-tetrahydro-1<i>H</i>-benzazepines and Related Compounds

Hidenori Ogawa, Hiroshi Yamashita, Kazumi Kondo et al. · Journal of Medicinal Chemistry · 1996 · 87 citations · Full text

, , +8