Characterization of histamine H2-receptors in human neutrophils with a series of guanidine analogues of impromidine

Definition and Antagonism of Histamine H2-receptors

J. W. Black, W. A. M. Duncan, C. J. DURANT et al. · Nature · 1972 · 2.3K citations

Medicine, Medicinal Chemistry, Pharmacology +12

Highly potent and selective ligands for histamine H3-receptors

J.M. Arrang, M. Garbarg, J.-C. Lancelo et al. · Nature · 1987 · 902 citations

Medicine, Medicinal Chemistry, Pharmacology +15

pA, A NEW SCALE FOR THE MEASUREMENT OF DRUG ANTAGONISM

H. O. Schild · British Journal of Pharmacology and Chemotherapy · 1947 · 759 citations · Full text

Medicine, Pharmacology, Comparative Pharmacology +10

Dimaprit-[S-[3-(N,N-dimethylamino)propyl]isothiourea] —A highly specific histamine H2-receptor agonist. Part 1. Pharmacology

Michael E. Parsons, D. A. A. Owen, C. Robin Ganellin et al. · Inflammation Research · 1977 · 241 citations

Medicine, Medicinal Chemistry, Pharmacology +7

Impromidine (SK&F 92676) is a very potent and specific agonist for histamine H2 receptors

G. J. DURANT, W. A. M. Duncan, C. Robin Ganellin et al. · Nature · 1978 · 222 citations

Medicine, Pharmacology, Pharmacodynamics +7