Concepedia

Biochemical characterization of desloratadine, a potent antagonist of the human histamine H1 receptor

John C. Anthes, Helen Gilchrest, Christian Richard, Stephen Eckel, Robert E. West, Shirley M. Williams, Scott Greenfeder, Motasim Billah, William Kreutner, Robert W. Egan

European Journal of Pharmacology · 2002 · 120 citations · 28 references

DOI

Concepts

References

28

Relationship between the inhibition constant (KI) and the concentration of inhibitor which causes 50 per cent inhibition (I50) of an enzymatic reaction

Yung-Chi Cheng, William H. Prusoff · Biochemical Pharmacology · 1973 · 12.9K citations

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Cloning and Functional Expression of the Human Histamine H<sub>3</sub>Receptor

Timothy W. Lovenberg, Barbara Roland, Sandy J. Wilson et al. · Molecular Pharmacology · 1999 · 700 citations · Full text

, , +16

Mechanism of the Cardiotoxic Actions of Terfenadine

Raymond L. Woosley · JAMA · 1993 · 617 citations

, , +14

Molecular Cloning and Characterization of a Novel Type of Histamine Receptor Preferentially Expressed in Leukocytes

Tamaki Oda, Noriyuki Morikawa, Yoko Saito et al. · Journal of Biological Chemistry · 2000 · 613 citations · Full text

, , +14

Torsades de pointes occurring in association with terfenadine use

B. P. Monahan · JAMA · 1990 · 554 citations

, , +13