Concepedia

Design and synthesis of N6-substituted-4′-thioadenosine-5′-uronamides as potent and selective human A3 adenosine receptor agonists

Won Jun Choi, Hyuk Woo Lee, Hea Ok Kim, Moshe Chinn, Zhan‐Guo Gao, Amit R. Patel, Kenneth A. Jacobson, Hyung Ryong Moon, Young Hoon Jung, Lak Shin Jeong

Bioorganic & Medicinal Chemistry · 2009 · 19 citations · 13 references

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13

Structure-Activity Relationships of N6-Benzyladenosine-5'-uronamides as A3-Selective Adenosine Agonists

Carola Gallo‐Rodriguez, Xiao-duo Ji, Neli Melman et al. · Journal of Medicinal Chemistry · 1994 · 238 citations · Full text

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2-Substitution of N6-Benzyladenosine-5'-uronamides Enhances Selectivity for A3 Adenosine Receptors

Hea O. Kim, Xiao-duo Ji, Suhaib M. Siddiqi et al. · Journal of Medicinal Chemistry · 1994 · 204 citations · Full text

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A physiological role of the adenosine A <sub>3</sub> receptor: Sustained cardioprotection

Bruce T. Liang, Kenneth A. Jacobson · Proceedings of the National Academy of Sciences · 1998 · 201 citations · Full text

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Structural Determinants of A<sub>3</sub> Adenosine Receptor Activation:  Nucleoside Ligands at the Agonist/Antagonist Boundary

Zhan‐Guo Gao, Soo‐Kyung Kim, Thibaud Biadatti et al. · Journal of Medicinal Chemistry · 2002 · 137 citations · Full text

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N6-Substituted adenosine derivatives: selectivity, efficacy, and species differences at A3 adenosine receptors

Zhan‐Guo Gao, Joshua B. Blaustein, Ariel S. Gross et al. · Biochemical Pharmacology · 2003 · 134 citations

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