Diastereoselective reduction of β-ketophosphonates derived from amino acids. A new entry to enantiopure β-hydroxy-γ-aminophosphonate derivatives

Phosphinic Acid Analogs of GABA. 1. New Potent and Selective GABAB Agonists

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Medicine, Medicinal Chemistry, Pharmacology +13

Preparation of fluoro- and hydroxy-4-(phosphonomethyl)-D,L-phenylalanine suitably protected for solid-phase synthesis of peptides containing hydrolytically stable analogs of O-phosphotyrosine

Terrence R. Burke, Mark S. Smyth, Motoyoshi Nomizu et al. · The Journal of Organic Chemistry · 1993 · 162 citations

Natural Sciences, Biochemistry, Chemistry +10

The Catalytic Asymmetric Aminohydroxylation of Unsaturated Phosphonates

Allen A. Thomas, K. Barry Sharpless · The Journal of Organic Chemistry · 1999 · 123 citations

Pharmacy, Biochemistry, Chemistry +6

Synthesis of monofluoro- and difluoro- methylenephosphonate analogues of sn-glycerol-3-phosphate as substrates for glycerol-3-phosphate dehydrogenase and the X-ray structure of the fluoromethylenephosphonate moiety

Jens Nieschalk, Andrei S. Batsanov, David O’Hagan et al. · Tetrahedron · 1996 · 111 citations

Life Sciences, Biochemistry, Biology +9

New inhibitors of renin that contain novel phosphostatine Leu-Val replacements

Joseph F. Dellaria, Robert G. Maki, Herman H. Stein et al. · Journal of Medicinal Chemistry · 1990 · 103 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +11