Synthetic Communications · 2003 · 12 citations · 35 references
Natural SciencesChemistryMedicinal ChemistryOrganic ChemistrySynthetic Medicinal ChemistryHeterocycle SynthesisHeterocyclic ChemistryOrganic SynthesisOxazole ChemistryOxazole SynthesisSteric Constraints
Abstract Optimized conditions for the preparation of 4-ethoxyalkyliden-5(4H)-oxazolones were developed. A considerable steric hindrance was observed on the nucleophilic substitution of the ethoxy group by amines.
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Didehydroamino Acids (DDAA) and Didehydropeptides (DDP)
Ulrich Schmidt, Albrecht Lieberknecht, Jochen Wild · Synthesis · 1988 · 202 citations