Concepedia

Melatonin-mediated regulation of human MT1 melatonin receptors expressed in mammalian cells

Matthew J. Gerdin, Monica I. Masana, Margarita L. Dubocovich

Biochemical Pharmacology · 2004 · 80 citations · 28 references

DOI

Concepts

References

28

Relationship between the inhibition constant (KI) and the concentration of inhibitor which causes 50 per cent inhibition (I50) of an enzymatic reaction

Yung-Chi Cheng, William H. Prusoff · Biochemical Pharmacology · 1973 · 12.9K citations

, , +14

Cloning and characterization of a mammalian melatonin receptor that mediates reproductive and circadian responses

Steven M. Reppert, David R. Weaver, Takashi Ebisawa · Neuron · 1994 · 1.1K citations · Full text

, , +14

Molecular Dissection of Two Distinct Actions of Melatonin on the Suprachiasmatic Circadian Clock

Chen Liu, David R. Weaver, Xiaowei Jin et al. · Neuron · 1997 · 719 citations · Full text

, , +15

Selective MT <sub>2</sub> melatonin receptor antagonists block melatonin‐mediated phase advances of circadian rhythms

Margarita L. Dubocovich, Kenneth Yun, Walid M. Al‐Ghoul et al. · The FASEB Journal · 1998 · 362 citations

, , +17

Structural Instability of a Constitutively Active G Protein-coupled Receptor

Ulrik Gether, Roland Seifert, Juan Antonio Ballesteros‐Cánovas et al. · Journal of Biological Chemistry · 1997 · 299 citations · Full text

, , +17