Fluorinated azines and benzazines containing oxygen or sulfur atoms

ENZYMES AT WORK

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Engineering, Altmetric Attention Score, Enzymatic Modification +17

2-Amino-4<i>H</i>-3,1-benzoxazin-4-ones as Inhibitors of C1r Serine Protease

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Combinatorial Chemistry, Complement Enzyme C1r, Medicinal Chemistry +14

Atropisomeric quinazolin-4-one derivatives are potent noncompetitive α-amino-3-hydroxy-5-methyl-4-isoxazolepropionic acid (AMPA) receptor antagonists

W. M. WELCH, Frank E. Ewing, J. HUANG et al. · Bioorganic & Medicinal Chemistry Letters · 2001 · 123 citations

Molecular Pharmacology, Biochemistry, Atropisomeric Quinazolin-4-one Derivatives +7

Catalytic, Asymmetric Synthesis of 1,4‐Benzoxazinones: A Remarkably Enantioselective Route to α‐Amino Acid Derivatives from <i>o</i>‐Benzoquinone Imides

Jamison Wolfer, Tefsit Bekele, Ciby J. Abraham et al. · Angewandte Chemie International Edition · 2006 · 100 citations

O-benzoquinone Imides, Catalytic Asymmetric Synthesis, Enantioselective Route +16

Mammalian topoisomerase II inhibitory activity of 1-cyclopropyl-6,8-difluoro-1,4-dihydro-7-(2,6-dimethyl-4-pyridinyl)-4-oxo-3-quinolinecarboxylic acid and related derivatives

Mark P. Wentland, George Y. Lesher, Michael Reuman et al. · Journal of Medicinal Chemistry · 1993 · 73 citations · Full text