Concepedia

Synthesis and SAR studies of 1,4-diazabicyclo[3.2.2]nonane phenyl carbamates – subtype selective, high affinity α7 nicotinic acetylcholine receptor agonists

Christopher J. O’Donnell, Langu Peng, Brian T. O’Neill, Eric P. Arnold, Robert J. Mather, Steven B. Sands, Alka Shrikhande, Lorraine A. Lebel, Douglas K. Spracklin, Frank M. Nedza

Bioorganic & Medicinal Chemistry Letters · 2009 · 15 citations · 20 references

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Concepts

References

20

Palladium(0)-Catalyzed Cross-Coupling Reaction of Alkoxydiboron with Haloarenes: A Direct Procedure for Arylboronic Esters

Tatsuo Ishiyama, Miki Murata, Norio Miyaura · The Journal of Organic Chemistry · 1995 · 1.6K citations

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Association of Promoter Variants in the α7 Nicotinic Acetylcholine Receptor Subunit Gene With an Inhibitory Deficit Found in Schizophrenia

Sherry Leonard, Judith Gault, Jan Hopkins et al. · Archives of General Psychiatry · 2002 · 442 citations

, , +15

Pharmacological characterization of recombinant human neuronal nicotinic acetylcholine receptors h alpha 2 beta 2, h alpha 2 beta 4, h alpha 3 beta 2, h alpha 3 beta 4, h alpha 4 beta 2, h alpha 4 beta 4 and h alpha 7 expressed in Xenopus oocytes.

Laura E. Chavez-Noriega, James H. Crona, Mark Washburn et al. · PubMed · 1997 · 393 citations

, , +17

SSR180711, a Novel Selective α7 Nicotinic Receptor Partial Agonist: (II) Efficacy in Experimental Models Predictive of Activity Against Cognitive Symptoms of Schizophrenia

Philippe Pichat, Olivier Bergis, Jean-Paul Terranova et al. · Neuropsychopharmacology · 2006 · 237 citations

, , +13

Pharmacological Characterization of Recombinant Human Neuronal Nicotinic Acetylcholine Receptors hα2β2, hα2β4, hα3β2, hα3β4, hα4β2, hα4β4 and hα7 Expressed in Xenopus Oocytes

Laura E. Chavez-Noriega, James H. Crona, Mark Washburn et al. · Journal of Pharmacology and Experimental Therapeutics · 1997 · 206 citations

, , +14