Concepedia

The Peptides Mimicking the Third Intracellular Loop of 5-Hydroxytryptamine Receptors of the Types 1B and 6 Selectively Activate G Proteins and Receptor-Specifically Inhibit Serotonin Signaling via the Adenylyl Cyclase System

I. I. Tarasenko, Gennady P. Vlasov

International Journal of Peptide Research and Therapeutics · 2010 · 63 citations · 37 references

DOI

Concepts

References

37

G‐protein‐coupled receptors: molecular mechanisms involved in receptor activation and selectivity of G‐protein recognition

Jürgen Wess · The FASEB Journal · 1997 · 592 citations

, , +19

Activation and inhibition of G protein-coupled receptors by cell-penetrating membrane-tethered peptides

Lidija Covic, Amy L. Gresser, Joyce R. Talavera et al. · Proceedings of the National Academy of Sciences · 2002 · 312 citations · Full text

Pepducin-based intervention of thrombin-receptor signaling and systemic platelet activation

Lidija Covic, Meghna V. Misra, Jehangir Badar et al. · Nature Medicine · 2002 · 277 citations

, , +9

Synthetic peptides as probes for G protein function. Carboxyl-terminal G alpha s peptides mimic Gs and evoke high affinity agonist binding to beta-adrenergic receptors.

Mark M. Rasenick, Masayuki Watanabe, Milenko Lazarevic et al. · Journal of Biological Chemistry · 1994 · 130 citations · Full text

The G Protein β Subunit Is a Determinant in the Coupling of Gs to the β1-Adrenergic and A2a Adenosine Receptors

William E. McIntire, Gavin MacCleery, James C. Garrison · Journal of Biological Chemistry · 2001 · 102 citations · Full text