Differential inhibition of murine Bcrp1/Abcg2 and human BCRP/ABCG2 by the mycotoxin fumitremorgin C

Rapid colorimetric assay for cellular growth and survival: Application to proliferation and cytotoxicity assays

Tim R. Mosmann · Journal of Immunological Methods · 1983 · 55.6K citations

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Potent and specific inhibition of the breast cancer resistance protein multidrug transporter in vitro and in mouse intestine by a novel analogue of fumitremorgin C.

Arnold van Loevezijn, Jeany M Lakhai, Martin van der Valk et al. · PubMed · 2002 · 687 citations

Medicine, Medicinal Chemistry, Pharmacology +17

Fumitremorgin C reverses multidrug resistance in cells transfected with the breast cancer resistance protein.

Sridhar K. Rabindran, D D Ross, L. Austin Doyle et al. · PubMed · 2000 · 490 citations

Medicine, Oncology, Pharmacology +16

Pheophorbide a Is a Specific Probe for ABCG2 Function and Inhibition

Robert W. Robey, Kenneth Steadman, Orsolya Polgár et al. · Cancer Research · 2004 · 355 citations · Full text

Life Sciences, Cell Biology, Pharmacology +17

The mouse Bcrp1/Mxr/Abcp gene: amplification and overexpression in cell lines selected for resistance to topotecan, mitoxantrone, or doxorubicin.

John Allen, R F Brinkhuis, Jan Wijnholds et al. · PubMed · 1999 · 352 citations

Medicine, Oncology, Pharmacology +17