Concepedia

Loss of antagonistic activity of tamoxifen by replacement of one N-methyl of its side chain by fluorinated residues

Vangelis Agouridas, Ioanna Laı ̈os, Anny Cleeren, Elyane Kizilian, Emmanuel Magnier, Jean‐Claude Blazejewski, Guy Leclercq

Bioorganic & Medicinal Chemistry · 2006 · 22 citations · 24 references

DOI

Concepts

References

24

Molecular basis of agonism and antagonism in the oestrogen receptor

A.M. Brzozowski, A.C.W. Pike, Zbigniew Dauter et al. · Nature · 1997 · 3.3K citations

, , +14

Cyanohydridoborate anion as a selective reducing agent

Richard F. Borch, Mark D. Bernstein, H. D. Durst · Journal of the American Chemical Society · 1971 · 1.8K citations

, , +5

Correlation of the Base Strengths of Amines<sup>1</sup>

H. K. Hall · Journal of the American Chemical Society · 1957 · 793 citations

, , +8

The 26S Proteasome Is Required for Estrogen Receptor-α and Coactivator Turnover and for Efficient Estrogen Receptor-α Transactivation

David M. Lonard, Zafar Nawaz, Carolyn L. Smith et al. · Molecular Cell · 2000 · 557 citations · Full text

, , +15

Forty years of hydride reductions

Herbert C. Brown, S. Krishnamurthy · Tetrahedron · 1979 · 449 citations

, , +4