Concepedia

The development of first Staphylococcus aureus SplB protease inhibitors: Phosphonic analogues of glutamine

Ewa Burchacka, Maciej Walczak, Marcin Sieńczyk, Grzegorz Dubin, Michal Zdzalik, Potempa Jan, Józef Oleksyszyn

Bioorganic & Medicinal Chemistry Letters · 2012 · 26 citations · 15 references

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15

On the size of the active site in proteases. I. Papain

Israël Schechter, Arieh Berger · Biochemical and Biophysical Research Communications · 1967 · 5.2K citations

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Irreversible inhibition of serine proteases by peptide derivatives of (.alpha.-aminoalkyl)phosphonate diphenyl esters

Józef Oleksyszyn, James C. Powers · Biochemistry · 1991 · 198 citations

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Irreversible Inhibition of Serine Proteases – Design and In Vivo Activity of Diaryl α-Aminophosphonate Derivatives

Marcin Sieńczyk, Józef Oleksyszyn · Current Medicinal Chemistry · 2009 · 145 citations

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Molecular Characterization of a Novel<i>Staphylococcus aureus</i>Serine Protease Operon

Samantha B. Reed, Carla A. Wesson, Linda E. Liou et al. · Infection and Immunity · 2001 · 136 citations · Full text

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Novel amidine-containing peptidyl phosphonates as irreversible inhibitors for blood coagulation and related serine proteases

Józef Oleksyszyn, Bogdan Boduszek, Chih-Min Kam et al. · Journal of Medicinal Chemistry · 1994 · 99 citations

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