Synthesis and cytotoxic evaluation of thiourea and N-bis-benzothiazole derivatives: A novel class of cytotoxic agents

Parallel Synthesis of a Library of Benzoxazoles and Benzothiazoles Using Ligand-Accelerated Copper-Catalyzed Cyclizations of <i>ortho</i>-Halobenzanilides

Ghotas Evindar, Robert A. Batey · The Journal of Organic Chemistry · 2006 · 482 citations

Natural Sciences, Chemistry, Medicinal Chemistry +17

Antitumor Benzothiazoles. 26. 2-(3,4-Dimethoxyphenyl)-5-fluorobenzothiazole (GW 610, NSC 721648), a Simple Fluorinated 2-Arylbenzothiazole, Shows Potent and Selective Inhibitory Activity against Lung, Colon, and Breast Cancer Cell Lines

Catriona G. Mortimer, Geoffrey Wells, Jean-Philippe Crochard et al. · Journal of Medicinal Chemistry · 2005 · 474 citations

Medicine, Medicinal Chemistry, Pharmacology +11

Antitumor Benzothiazoles. 16. Synthesis and Pharmaceutical Properties of Antitumor 2-(4-Aminophenyl)benzothiazole Amino Acid Prodrugs

Ian Hutchinson, S. A. Jennings, B. Rao Vishnuvajjala et al. · Journal of Medicinal Chemistry · 2001 · 420 citations

Pharmacy, Medicinal Chemistry, Pharmacology +15

Synthesis and antimicrobial activity of some new thiazole, thiophene and pyrazole derivatives containing benzothiazole moiety

Samir Bondock, Walid Fadaly, M. A. Metwally · European Journal of Medicinal Chemistry · 2010 · 391 citations

Pharmacy, Chemistry, Medicinal Chemistry +14

Palladium-Catalyzed Synthesis of 2-Substituted Benzothiazoles via a C−H Functionalization/Intramolecular C−S Bond Formation Process

Kiyofumi Inamoto, Chisa Hasegawa, Kou Hiroya et al. · Organic Letters · 2008 · 286 citations

Natural Sciences, Chemistry, Catalysis +15