MedChemComm · 2014 · 12 citations · 37 references
PharmacyMedicinal ChemistryPharmacologyBioisosterismCancer PharmacologyDrug DiscoveryHeterocyclic Chemistry
The diazo functionality of the kinamycins may not be an absolute requirement for bioactivity.
37
Modern physical organic chemistry
Choice Reviews Online · 2006 · 2.4K citations
Bioactivation as a Model for Drug Design Bioreductive Alkylation
Harold W. Moore · Science · 1977 · 433 citations