Concepedia

The discovery of non-benzimidazole and brain-penetrant prolylcarboxypeptidase inhibitors

Thomas H. Graham, Hong C. Shen, Wensheng Liu, Yusheng Xiong, Andreas Verras, Kelly Bleasby, Urmi R. Bhatt, Renee M. Chabin, Dunlu Chen, Qing Chen,

Bioorganic & Medicinal Chemistry Letters · 2011 · 16 citations · 27 references

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References

27

Structure–activity relationship of P-glycoprotein substrates and modifiers

Anna Seelig, Ewa Landwojtowicz · European Journal of Pharmaceutical Sciences · 2000 · 277 citations

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Transport of small molecules through the blood-brain barrier: biology and methodology

William M. Pardridge · Advanced Drug Delivery Reviews · 1995 · 274 citations

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Classification Analysis of P-Glycoprotein Substrate Specificity

Remigijus Didžiapetris, Pranas Japertas, Alex Avdeef et al. · Journal of drug targeting · 2003 · 256 citations

, , +15

Identification and Characterization of Prolylcarboxypeptidase as an Endothelial Cell Prekallikrein Activator

Zia Shariat‐Madar, Fakhri Mahdi, Alvin H. Schmaier · Journal of Biological Chemistry · 2002 · 255 citations · Full text

, , +14

Trifluoromethyl group: an effective xenobiotic function for peptide backbone modification

Matteo Zanda · New Journal of Chemistry · 2004 · 162 citations

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