Concepedia

Quantitative structure-agonist activity relationship of capsaicin analogues

Gilles Klopman, Ju-Yun Li

Journal of Computer-Aided Molecular Design · 1995 · 26 citations · 34 references

DOI

Concepts

References

34

Structure and energetics of ligand binding to proteins: <i>Escherichia coli</i> dihydrofolate reductase‐trimethoprim, a drug‐receptor system

Pnina Dauber‐Osguthorpe, Victoria A. Roberts, David J. Osguthorpe et al. · Proteins Structure Function and Bioinformatics · 1988 · 2.1K citations

, , +16

Capsazepine: a competitive antagonist of the sensory neurone excitant capsaicin

Stuart Bevan, Sandeep S Hothi, Glyn A. Hughes et al. · British Journal of Pharmacology · 1992 · 584 citations · Full text

, , +16

Capsaicin-induced ion fluxes in dorsal root ganglion cells in culture

JN Wood, J. Winter, I. F. James et al. · Journal of Neuroscience · 1988 · 566 citations · Full text

, , +17

Resiniferatoxin, a phorbol-related diterpene, acts as an ultrapotent analog of capsaicin, the irritant constituent in red pepper

A Szállaśi, Peter M. Blumberg · Neuroscience · 1989 · 437 citations · Full text

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Hydrophobicity and Central Nervous System Agents: On the Principle of Minimal Hydrophobicity in Drug Design

Corwin Hansch, J.P. Björkroth, Albert J. Leo · Journal of Pharmaceutical Sciences · 1987 · 435 citations

, , +14