Binding of the bidentate inhibitor [3H]HACBO-Gly to the rat brain neutral endopeptidase “enkephalinase”

Design of potent competitive inhibitors of angiotensin-converting enzyme. Carboxyalkanoyl and mercaptoalkanoyl amino acids

David W. Cushman, H.S. Cheung, Emily F. Sabo et al. · Biochemistry · 1977 · 901 citations

Pharmacy, Medicinal Chemistry, Pharmacology +10

The enkephalinase inhibitor thiorphan shows antinociceptive activity in mice

B P Roques, M C Fournié-Zaluski, E. Soroca et al. · Nature · 1980 · 707 citations

Medicine, Neuroscience, Pharmacology +10

High-affinity enkephalin-degrading peptidase in brain is increased after morphine

Bernard Malfroy, Jean-Paul Swerts, Anne Guyon et al. · Nature · 1978 · 650 citations

Medicine, Neuroscience, Pharmacology +12

The purification and specificity of a neutral endopeptidase from rabbit kidney brush border

M. A. Kerr, A J Kenny · Biochemical Journal · 1974 · 462 citations · Full text

Life Sciences, Biochemistry, Molecular Biology +17

Analgesic effects of kelatorphan, a new highly potent inhibitor of multiple enkephalin degrading enzymes

Marie‐Claude Fournié‐Zaluski, Pierre Chaillet, Romaine Bouboutou et al. · European Journal of Pharmacology · 1984 · 167 citations

Medicine, Medicinal Chemistry, Pharmacology +11