Interaction of anisatin with rat brain γ-aminobutyric acida receptors: allosteric modulation by competitive antagonists

A point mutation in a Drosophila GABA receptor confers insecticide resistance

Richard H. ffrench‐Constant, Thomas A. Rocheleau, J.C. Steichen et al. · Nature · 1993 · 582 citations

Biology, Genetics, Entomology +10

[35S]t-butylbicyclophosphorothionate binds with high affinity to brain-specific sites coupled to gamma-aminobutyric acid-A and ion recognition sites.

Richard F. Squires, John E. Casida, Michael Richardson et al. · Molecular Pharmacology · 1983 · 552 citations

Molecular Pharmacology, Biochemistry, Medicine +10

GABA, Bicuculline and Central Inhibition

D.R. Curtis, A.W. Duggan, D. Felix et al. · Nature · 1970 · 539 citations

Medicine, Mechanism Of Action, Neuropharmacology +7

Bicuculline and Gabazine Are Allosteric Inhibitors of Channel Opening of the GABA_AReceptor

Shinya Ueno, John Bracamontes, Chuck Zorumski et al. · Journal of Neuroscience · 1997 · 259 citations · Full text

Gaba-binding Site, Anesthetic Mechanism, Pharmacotherapy +22

Interaction of picrotoxin with GABAA receptor channel-lining residues probed in cysteine mutants

Ming Xu, Douglas F. Covey, Myles H. Akabas · Biophysical Journal · 1995 · 145 citations · Full text