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Discovery of potent, selective and orally bioavailable triaryl-sulfonamide based PTP1B inhibitors

Dipam Patel, Mukul R. Jain, Shailesh R. Shah, Rajesh Bahekar, Pradip Jadav, Amit Joharapurkar, Nirav Dhanesha, Mubeen Shaikh, K Sairam, Prashant B. Kapadnis

Bioorganic & Medicinal Chemistry Letters · 2011 · 43 citations · 17 references

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Global Prevalence of Diabetes

Sarah H. Wild, Gojka Roglić, Anders Green et al. · Diabetes Care · 2004 · 15.3K citations

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Oral Antidiabetic Agents

Andrew J. Krentz, Clifford J. Bailey · Drugs · 2005 · 1.1K citations

Identification of a second aryl phosphate-binding site in protein-tyrosine phosphatase 1B: A paradigm for inhibitor design

Yoram A. Puius, Yu Zhao, Michael Sullivan et al. · Proceedings of the National Academy of Sciences · 1997 · 402 citations

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Recent Advances in the Discovery of Competitive Protein Tyrosine Phosphatase 1B Inhibitors for the Treatment of Diabetes, Obesity, and Cancer

Andrew P. Combs · Journal of Medicinal Chemistry · 2009 · 316 citations · Full text

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Development and Characterization of a Glucagon-Like Peptide 1-Albumin Conjugate

Jung‐Guk Kim, Laurie L. Baggio, Dominique Bridon et al. · Diabetes · 2003 · 212 citations

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