Bioorganic & Medicinal Chemistry · 2007 · 41 citations · 10 references
PharmacyMedicinal ChemistryPharmacologyDrug DesignDrug DiscoveryEnzymologyEnzyme InhibitionNatural Product-based Drug DesignPotency OptimizationChemical Synthesis Of AnaloguesEnzyme Inhibitor SynthesisInhibitor ScreeningMechanism-based InhibitorsMedicinal Chemistry Applications
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A metalloproteinase disintegrin that releases tumour-necrosis factor-α from cells
Roy A. Black, Charles T. Rauch, Carl J. Kozlosky et al. · Nature · 1997 · 3.1K citations