Synthesis and evaluation of fluoro substituted pyridinylcarboxamides and their phenylazo analogues for potential dopamine D3 receptor PET imaging

Molecular cloning and characterization of a novel dopamine receptor (D3) as a target for neuroleptics

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Life Sciences, Neuroscience, Pharmacology +12

Selective inhibition of cocaine-seeking behaviour by a partial dopamine D3 receptor agonist

Maria Pilla, Sylvie Perachon, François Sautel et al. · Nature · 1999 · 568 citations

Medicine, Neuroscience, Pharmacology +13

Radiosynthesis and Evaluation of [¹¹C]-(+)-4-Propyl-3,4,4a,5,6,10b-hexahydro-2<i>H</i>-naphtho[1,2-<i>b</i>][1,4]oxazin-9-ol as a Potential Radiotracer for in Vivo Imaging of the Dopamine D2 High-Affinity State with Positron Emission Tomography

Alan A. Wilson, Patrick N. McCormick, Shitij Kapur et al. · Journal of Medicinal Chemistry · 2005 · 226 citations

Medicine, Nuclear Medicine, Pharmacology +17

Interactive SAR Studies:  Rational Discovery of Super-Potent and Highly Selective Dopamine D3 Receptor Antagonists and Partial Agonists

Laura Bettinetti, Karin Schlotter, Harald Hübner et al. · Journal of Medicinal Chemistry · 2002 · 194 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +17

Conjugated Enynes as Nonaromatic Catechol Bioisosteres:  Synthesis, Binding Experiments, and Computational Studies of Novel Dopamine Receptor Agonists Recognizing Preferentially the D₃Subtype

Harald Hübner, Christian Haubmann, Wolfgang Utz et al. · Journal of Medicinal Chemistry · 2000 · 168 citations · Full text

Medicine, Medicinal Chemistry, Pharmacology +17