Concepedia

Characterization of opiates, neuroleptics, and synthetic analogs at ORL1 and opioid receptors

Nurulain T. Zaveri, Willma E. Polgar, Cris M Olsen, A B Kelson, Peter Grundt, John W. Lewis, Lawrence Toll

European Journal of Pharmacology · 2001 · 59 citations · 26 references

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26

Relationship between the inhibition constant (KI) and the concentration of inhibitor which causes 50 per cent inhibition (I50) of an enzymatic reaction

Yung-Chi Cheng, William H. Prusoff · Biochemical Pharmacology · 1973 · 12.9K citations

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Modulation by mu-opioid agonists of guanosine-5'-O-(3-[35S]thio)triphosphate binding to membranes from human neuroblastoma SH-SY5Y cells.

John R. Traynor, Stefan R. Nahorski · Molecular Pharmacology · 1995 · 462 citations

, , +17

Narcotic antagonists in the benzomorphan series

LouisS. Harris · Naunyn-Schmiedeberg s Archives of Pharmacology · 1964 · 321 citations

, , +6

A synthetic agonist at the orphanin FQ/nociceptin receptor ORL1: Anxiolytic profile in the rat

François Jenck, Juergen Wichmann, Frank M. Dautzenberg et al. · Proceedings of the National Academy of Sciences · 2000 · 274 citations

, , +14

A new selective antagonist of the nociceptin receptor

Remo Guerrini, Girolamo Calò, Anna Rizzi et al. · British Journal of Pharmacology · 1998 · 241 citations · Full text

, , +13