A convenient synthesis of N-protected diphenyl phosphonate ester analogues of ornithine, lysine and homolysine.

Fast and selective oxidation of primary alcohols to aldehydes or to carboxylic acids and of secondary alcohols to ketones mediated by oxoammonium salts under two-phase conditions

Pier Lucio Anelli, Carlo Biffi, Fernando Montanari et al. · The Journal of Organic Chemistry · 1987 · 772 citations

Natural Sciences, Chemistry, Biocatalysis +10

1-Aminoalkylphosphonous acids. Part 1. Isosteres of the protein amino acids

E. K. Baylis, Colin D. Campbell, John G. Dingwall · Journal of the Chemical Society Perkin Transactions 1 · 1984 · 344 citations

Life Sciences, Biochemistry, Chemistry +11

Direct determination of the protonation states of aspartic acid-102 and histidine-57 in the tetrahedral intermediate of the serine proteases: neutron structure of trypsin

Anthony A. Kossiakoff, Steven A. Spencer · Biochemistry · 1981 · 266 citations

Life Sciences, Biochemistry, Chemistry +17

Irreversible inhibition of serine proteases by peptide derivatives of (.alpha.-aminoalkyl)phosphonate diphenyl esters

Józef Oleksyszyn, James C. Powers · Biochemistry · 1991 · 198 citations

Life Sciences, Biochemistry, Pharmacology +15

CCCXII.—A modification of the Gabriel synthesis of amines

H. R. Ing, Richard H. F. Manske · Journal of the Chemical Society (Resumed) · 1926 · 194 citations

Natural Sciences, Chemistry, Organic Chemistry +1